释义 |
1 ?二氟甲基鸟氨酸 二氟甲基鸟氨酸(DFMO)和乙基乙二醛二眯腺(EGBG),是两种强效多胺合成阻断剂,分别抑制多胺合成途径中的限速酶鸟氨酸脱装酶和s一腺昔甲硫氨酸脱狡酶,由美... 2 ?二甲亚砜 ()其它正在研究的有关药物有: 过氧化酶增殖物活化受体配体二甲亚砜(DFMO)钙剂(结合胆酸)维生素D表皮生长因子受体抑制剂酪氨酸激酶抑制剂血管内皮生长因子抑制剂基质金属蛋白酶抑制剂等 3 ?抑制剂二氟甲基鸟氨酸 随后用ODC抑制剂二氟甲基鸟氨酸(difluoromethylornithine,DFMO)治疗,结果发现与未经治疗的糖尿病大鼠相比,治疗组大鼠的肾脏体积明显减小且肾小球滤过率(GFR)也出现... 4 ?二氟甲基鸟氨 (2)二氟甲基鸟氨(difluoromethylornithine,DFMO):又称依氟鸟氨酸(eflornithine),为一种鸟氨酸脱羧酶抑制剂,仅对冈比亚锥虫感染有效。
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Objective: To investigate the effects of DFMO on the growth characteristics, apoptosis and activity of telomerase of K562 cells. 目的研究二氟甲基鸟氨酸(DFMO)对K562细胞生长特性、凋亡及端粒酶活性的影响。 - 2
Conclusion: The growth inhibition and apoptosis induction of K562 cells treated by DFMO were associated with suppressed telomerase activity. 结论DFMO引起的K562细胞生长抑制及凋亡诱导与端粒酶活性抑制有关。 - 3
Meyskens says that DFMO, which is short for difluoromethylornithine, was developed as a cancer medication, but is now used to treat African sleeping sickness. Meyskens说,DFMO,α-二氟甲基鸟氨酸,是作为癌症治疗开发的,但现在用来治疗非洲昏睡病。
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