Objective: To study the antifungal activity of triazole alcohols by introduction of cyclopropyl as side chain.
目的：研究具有环丙基结构的三唑醇类化合物的抗真菌活性。
2
The key reactions included the formation of 9, 15-cyclopropyl function and double bond migration in the a ring to reestablish the GA skeleton.
本合成工作的关键为9,15环丙基的形成及在重建GA骨架时a环中双键的重排反应。
3
Moreover, we adopted an one - pot route combining the cyclopropanation and esterification of enoxysilane to prepare the cyclopropyl esters in moderate to good…